5-HT uptake & transport

Selective mGlu₈ receptor antagonist

Potent and selective 5-HT_2A receptor antagonist

Newly identified, highly selective FFA2-DREADD agonist

Selective P2Y₁ antagonist. Inhibits platelet aggregation.

Potent, selective P2Y₆ receptor antagonist

Potent, highly selective, non-competitive mGluR₅ antagonist

Invertebrate neurotransmitter. Chemogenetic DmOctβ1 receptor activator.

PAR₄ antagonist. Inhibits platelet aggregation.

TLR1/TLR2 agonist and potent NF-κB activator. Induces cytokine production.

Selective ERα estrogen receptor agonist