Receptors & Transporters

Estrogen receptor (ER) ligand.

D₂ receptor antagonist

Potent GLP-1 receptor agonist

Potent, selective, non-competitive mGlu₅ antagonist

Wnt/β-catenin inhibitor and PPARγ/δ antagonist.

Selective 5-HT uptake inhibitor. Affects differentiation of NSCs.

Selective glucocorticoid receptor agonist

Selective serotonin reuptake inhibitor and σ1 receptor agonist

Toll-like receptor 2 (TLR2) and TLR6 agonist

Selective PAR₂ peptide antagonist