Receptors & Transporters

Competitive, selective group 1 mGlu antagonist

Selective, non-competitive mGlu₁ antagonist

Potent, selective, non-competitive mGlu₅ antagonist

Potent, selective, non-competitive mGlu₁ antagonist

Potent, highly selective mGlu_1a antagonist. Water soluble.

Potent, highly selective mGlu_1a antagonist

Potent, selective mGluR₅ antagonist / mGluR₄ positive allosteric modulator

Potent, highly selective, non-competitive mGluR₅ antagonist

Potent, selective, non-competitive mGlu₁ antagonist