GluN2B

Non-selective purinergic P2X receptor antagonist

Potent and selective A_2A receptor antagonist

Potent, selective H₄ receptor silent antagonist

Potent, selective, non-competitive mGlu₁ antagonist

Selective 5-HT₂ receptor antagonist

Endogenous ionotropic glutamate / nicotinic antagonist.

Endogenous ionotropic glutamate / nicotinic antagonist. Sodium salt.

Selective, non-peptide AT₁ antagonist

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, potent, selective A₃AR covalent antagonist