Aurora kinase

Selective D₂-like receptor antagonist. Active enantiomer.

Standard D₂-like dopamine receptor antagonist

Selective, non-competitive AMPA / kainate receptor antagonist

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

Selective D₁-D₂ heteromer antagonist

TRPM2 antagonist. Cell permeable.

Potent, non-competitive GluN2A subunit selective NMDA receptor antagonist

Potent and selective orexin OX₂ antagonist

AT₁ antagonist and PPARγ partial agonist