Target

Novel, potent, selective A₃AR covalent antagonist

Potent, highly selective mGlu_1a antagonist. Water soluble.

Non-selective group I and II mGluR antagonist

Potent and selective 5-HT_2A receptor antagonist

Non-competitive NMDA receptor antagonist

Novel caged, fast-equilibrating glutamate receptor antagonist. Suitable for use as a synaptic probe.

Selective P2Y₁ antagonist. Inhibits platelet aggregation.

Potent, selective P2Y₆ receptor antagonist

Potent, highly selective, non-competitive mGluR₅ antagonist

Selective GluA2- lacking, Ca²⁺ permeable AMPA / kainate receptor antagonist