G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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  1. Olanzapine (HB1786)

    Description:

    5-HT2A and D2 antagonist. Potent DREADD agonist. Atypical antipsychotic.

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $54
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    Pack:
    50mg
    Price:
    $215
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  2. Description:

    LPA1 and LPA2 agonist. Inhibits differentiation of neural stem cells (NSCs) into neurons.

    Purity:

    >95%

    Pack:
    1mg
    Price:
    $70
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    Pack:
    5mg
    Price:
    $213
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  3. Pack:
    100mg
    Price:
    $86
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  4. Pack:
    100μg
    Price:
    $141
    Free trial
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    Pack:
    500μg
    Price:
    $348
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    Pack:
    1mg
    Price:
    $471
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  5. Pack:
    500μg
    Price:
    $182
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  6. Pack:
    1mg
    Price:
    $62
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    Pack:
    5mg
    Price:
    $95
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  7. P4pal10 (HB8677)

    Description:

    PAR4 antagonist. Inhibits platelet aggregation.

    Pack:
    1mg
    Price:
    $246
    Qty:
  8. Paliperidone (HB1798)

    Description:

    5-HT2A and D2 antagonist. Antipsychotic.

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $132
    Qty:
    Pack:
    50mg
    Price:
    $482
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  9. PD 102807 (HB1509)

    Description:

    Potent, selective M4 receptor antagonist. Promotes erythroid progenitors expansion.

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $287
    Qty:
  10. Perlapine (HB4889)

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    Description:

    Effective agonist for muscarinic-based DREADDs in vitro and in vivo. Non-CNO chemogenetic actuator

    Purity:

    >98%

    Pack:
    1mg
    Price:
    $33
    Qty:
    Pack:
    10mg
    Price:
    $132
    Qty:
    Pack:
    50mg
    Price:
    $545
    Qty:
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