G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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  1. Pack:
    50mg
    Price:
    $67
    Qty:
    Pack:
    250mg
    Price:
    $244
    Qty:
  2. LUF7445 (HB8439)

    Description:

    Novel, potent covalent A2A antagonist. Binds irreversibly.

    Pack:
    50μg
    Price:
    $275
    Qty:
  3. LUF7487 (HB9585)

    Description:

    Novel, covalent Affinity-Based Probe (AfBP). Clickable antagonist for the A2AR.

    Pack:
    50μg
    Price:
    $275
    Qty:
  4. Description:

    Novel, intracellular covalent chemokine CCR2 negative allosteric modulator (NAM). Binds irreversibly.

    Pack:
    50μg
    Price:
    $275
    Qty:
  5. LUF7602 (HB7286)

    Description:

    Novel, potent, selective A3AR covalent antagonist

    Pack:
    50μg
    Price:
    $275
    Qty:
  6. LUF7746 (HB6921)

    Description:

    The first covalent hA1AR partial agonist. Binds Irreversibly.

    Pack:
    50μg
    Price:
    $275
    Qty:
  7. Pack:
    50μg
    Price:
    $275
    Qty:
  8. Pack:
    50μg
    Price:
    $275
    Qty:
  9. LUF7982 (HB9905)

    Description:

    Novel Selective A2B covalent ligand. Binds irreversibly.

    Pack:
    50μg
    Price:
    $275
    Qty:
  10. Description:

    Potent, highly selective mGlu1a antagonist. Water soluble.

    Pack:
    10mg
    Price:
    $132
    Qty:
    Pack:
    50mg
    Price:
    $502
    Qty:
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