Receptors & Transporters

D₁-like receptor agonist

Potent, selective D₁-like receptor antagonist

Potent, selective, competitive GAT-1 GABA uptake inhibitor

Potent GABA_B receptor agonist

Selective glucagon receptor antagonist. Non-peptidic anti-diabetic agent

PAR₂ peptide agonist

Regulatory neuropeptide

Activates the hFFA2-DREADD

Selective mGlu₃ agonist, peptide neurotransmitter

Selective D₂-like receptor antagonist. 5-HT_2A antagonist.