Receptors & Transporters

Potent, selective 5-HT₇ receptor antagonist

Selective non-peptide orexin OX1 receptor antagonist

Potent 5-HT₆ antagonist

Potent, selective D₁-like receptor antagonist

Potent, selective D₁-like receptor antagonist

Selective D₂-like receptor antagonist. 5-HT_2A antagonist.

Mineralocorticoid and androgen receptor antagonist

Selective D₂-like receptor antagonist. Active enantiomer.

Standard D₂-like dopamine receptor antagonist

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).