Target

Potent mGlu₄ positive allosteric modulator

mGlu₄ positive allosteric modulator

Potent mGlu₅ positive allosteric modulator

Potent, selective ATP-competitive p38 MAPK inhibitor

Potent, selective p38α MAPK inhibitor

Calmodulin (CaM) antagonist

Potent 5-HT_1A receptor antagonist. D₄ receptor agonist.

Non-selective JAK3 inhibitor and potent EGFR inhibitor. Induces neural progenitor cell differentiation.

Potent tankyrase inhibitor. Wnt signaling inhibitor.

Potent, selective N-WASP inhibitor