Target

Potent, non-competitive GluN2A subunit selective NMDA receptor antagonist

Potent and selective orexin OX₂ antagonist

5-HT₄ partial agonist

AT₁ antagonist and PPARγ partial agonist

K_ir2.3 channel agonist

Acyl-CoA cholesterol acyltransferase 1 and 2 inhibitor

Antibacterial phytotoxin

Potent, specific, irreversible acetylcholinesterase (AChE) inhibitor.

Potent inward rectifier K⁺ channel blocker

Potent, selective K_ir1.1 channel blocker