Target

Guanosine analog with antiviral activity

Na⁺ channel blocker / glutamate inhibitor. TREK-1 K2P channel activator. Water soluble.

Na⁺ channel blocker

Na⁺ / Ca⁺ channel blocker

Reported to be a potent, selective Ca_v2.3 (R-type) channel blocker

Competitive EAAT blocker. Inhibits glutamate uptake.

Potent inward rectifier K⁺ channel blocker

Potent, selective K_ir1.1 channel blocker

Non-selective K⁺ channel blocker

Potent, selective, use-dependent Na⁺ channel blocker. Citrate free.