Target

Potent, selective PKA inhibitor

Novel, potent and selective GRK2/GRK3 inhibitor

Potent JAK inhibitor

Synthetic GP inhibitor

STAT3 inhibitor

Smo and hedgehog (Hh) signaling inhibitor. Also depletes stem like cancer cells and induces hESCs into endocrine cells.

Potent SERCA1a inhibitor

Potent calcineurin inhibitor. Inhibits MPTP opening.

Potent PP2B inhibitor

Transglutaminase inhibitor