Target

Endogenous ionotropic glutamate / nicotinic antagonist. Sodium salt.

Selective, non-peptide AT₁ antagonist

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, potent, selective A₃AR covalent antagonist

Potent, highly selective mGlu_1a antagonist. Water soluble.

5-HT_1D-preferring receptor antagonist

Potent, highly selective mGlu_1a antagonist

Non-selective group I and II mGluR antagonist

Non-selective group I/II mGluR antagonist

Non-selective group I and II mGluR antagonist. Water soluble sodium salt.