Target

D₁-like receptor agonist

Potent GABA_B receptor agonist

PAR₂ peptide agonist

Selective mGlu₃ agonist, peptide neurotransmitter

5-HT_1D, 5-HT_1B and 5-HT_1A receptor agonist

Abundant free amino acid found in the brain.

K_ir2.3 channel agonist

Potent, selective PPARγ agonist. Inhibits hematopoietic cell line growth.

Ultrapotent PSEM agonist for PSAM⁴-GlyR and PSAM⁴-5HT3. Brain penetrant.

Selective, ultrapotent PSEM agonist for PSAM⁴-GlyR and PSAM⁴-5HT3. Brain penetrant.