G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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Items 241-247 of 247

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  1. Description:

    Potent 5-HT3 antagonist and 5-HT4 agonist. Also selective IK1 channel agonist.

    Purity:

    >99%

    Pack:
    50mg
    Price:
    $615
    Qty:
  2. Description:

    5-HT2A and D2 antagonist. Atypical antipsychotic.

    Purity:

    >99%

    Pack:
    50mg
    Price:
    $575
    Qty:
  3. Pack:
    10mg
    Price:
    $130
    Qty:
    Pack:
    50mg
    Price:
    $540
    Qty:
  4. Zolmitriptan (HB1801)

    Description:

    Potent 5-HT1B/1D/1F agonist

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $103
    Qty:
    Pack:
    50mg
    Price:
    $349
    Qty:
  5. Zotepine (HB1778)

    Description:

    5-HT2A and dopamine D2 receptor antagonist. Atypical antipsychotic.

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $97
    Qty:
    Pack:
    50mg
    Price:
    $380
    Qty:
  6. Description:

    Histamine H1 antagonist. Potent actuator of a modified hM4Di "GRANPA" DREADD receptor.

    Purity:

    >99%

    Pack:
    500mg
    Price:
    $54
    Qty:
    Pack:
    1g
    Price:
    $75
    Qty:
  7. Pack:
    500μg
    Price:
    $141
    Qty:
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