Highly potent 5-HT3 receptor antagonist and 5-HT4 agonist (Ki values are 0.38 and 373 nM respectively). Also selective IK1 channel agonist. Shows anxiolytic and anti-emetic activity. Active in vivo.
Solubility & Handling
Solubility overview
Soluble in water (100mM) or DMSO (100mM)
Storage instructions
room temperature (desiccate)
Storage of solutions
Prepare and use solutions on the same day if possible. Store solutions at -20°C for up to one month if storage is required. Equilibrate to RT and ensure the solution is precipitate free before use.
Shipping Conditions
Stable for ambient temperature shipping. Follow storage instructions on receipt.
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.
Understanding purity and quality - a guide for life scientists