Receptors & Transporters

Selective, reverse mode Na⁺ / Ca²⁺ exchange inhibitor

Potent EGFR tyrosine kinase inhibitor

Inhibits α-MSH release inhibitors. Also increase dopamine levels.

L-aromatic amino acid decarboxylase inhibitor

5-HT and norepinephrine re-uptake inhibitor (SNRI)

Endogenous GLYT2 inhibitor / Ca_v3.1 / 3.2 / 3.3 current inhibitor

GLYT2 / GLYT2(EL2) inhibitor

LPA1 and LPA2 agonist. Inhibits differentiation of neural stem cells (NSCs) into neurons.

Potent, selective serotonin reuptake inhibitor. Selective GRK2 inhibitor.

FGFR1/ FGFR3 inhibitor. Inhibits oligodendrocyte progenitor proliferation and differentiation.