Target

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

Selective D₁-D₂ heteromer antagonist

GluK6-PSD-95 interaction inhibitor

TRPM2 antagonist. Cell permeable.

Abundant free amino acid found in the brain.

Competitive EAAT blocker. Inhibits glutamate uptake.

Selective class I HDAC inhibitor

Potent, selective Na_v1.7 inhibitor

Potent, non-competitive GluN2A subunit selective NMDA receptor antagonist

Potent and selective orexin OX₂ antagonist