Target

Selective leukotriene LTD4 receptor antagonist. Potent MRP1 inhibitor.

Potent, selective, non-competitive NMDA receptor antagonist

Less active enantiomer of (+)-MK 801. NMDA receptor antagonist.

Selective K_v7.2 / K_v7.4 channel activator

Selective mGlu₃ negative allosteric modulator

Selective K_2P2.1 (TREK-1) and K_2P10.1 (TREK-2) activator

Covalent K_2P2.1 (TREK-1) modulator. Used with CAT335 as part of the CATKLAMP chemogenetic strategy.

Selective K_2P2.1 (TREK-1) and K_2P10.1 (TREK-2) activator

Selective MLCK inhibitor

MAPKAPK2 (MK2) inhibitor. Cell permeable.