Target

Reversible trypsin-like and cysteine proteases inhibitor

K_ir6 channel activator

Potent and selective ACKR3 (CXCR7) agonist. Potentiates opioid peptide activity.

Highly potent, selective, competitive dipeptidyl-peptidase 4 inhibitor

K_v7 channel blocker

Potent MGMT inhibitor

Mitochondrial hexokinase inhibitor

Potent, selective µ-opioid receptor agonist

Potent and selective HIV-1 protease inhibitor

Selective, non-peptide AT₁ antagonist