Mineralocorticoid

Selective TGF-β signaling inhibitor. Induces cardiomyocyte differentiation in ESCs.

Selective, reverse mode Na⁺ / Ca²⁺ exchange inhibitor

Potent EGFR tyrosine kinase inhibitor

Potent and selective HIV-1 protease inhibitor

Potent endogenous MCH agonist

Inhibits α-MSH release inhibitors. Also increase dopamine levels.

L-aromatic amino acid decarboxylase inhibitor

5-HT and norepinephrine re-uptake inhibitor (SNRI)

Endogenous GLYT2 inhibitor / Ca_v3.1 / 3.2 / 3.3 current inhibitor

GLYT2 / GLYT2(EL2) inhibitor