Cannabinoid

Immediate precursor of dopamine

Potent, selective µ-opioid receptor agonist

The first covalent hA₁AR partial agonist. Binds Irreversibly.

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Novel, clickable Adenosine hA₃AR Affinity-Based Probe (AfBP).

Potent, selective group II receptor agonist

Selective H₁ receptor inverse agonist

5-HT₁/5-HT₂ antagonist. Shows affinity for 5-HT₆ and 5-HT₇.

Myelin oligodendrocyte glycoprotein fragment. Induces experimental multiple sclerosis-like disease.

Newly identified, highly selective FFA2-DREADD agonist