Receptors & Transporters

Selective, non-competitive mGlu₁ antagonist

Potent group III mGluR antagonist

Smo and hedgehog (Hh) signaling inhibitor. Also depletes stem like cancer cells and induces hESCs into endocrine cells.

Potent Formyl peptide receptor (FPR) inhibitor

Non-selective 5HT₂ antagonist

mGlu_1α / mGlu_5a agonist

TGF-βRI and CK1 inhibitor

Orphan nuclear receptor DAF-12 ligand

Estrogen receptors (ER) agonist. Phytoestrogen.

Potent, selective μ-opioid receptor agonist