Receptors & Transporters

Selective PAR₂ peptide antagonist

5-HT_2A receptor antagonist

Dopamine receptor antagonist with partial D₂-like selectivity

Estrogen receptor (ER) antagonist and high affinity GPER agonist

Potent and selective A_2A receptor antagonist

Potent, selective H₄ receptor silent antagonist

Potent, selective, non-competitive mGlu₁ antagonist

Selective 5-HT₂ receptor antagonist

Selective, non-peptide AT₁ antagonist

Novel, potent covalent A_2A antagonist. Binds irreversibly.