Target

Selective, non-competitive mGlu₁ antagonist

Potent, selective, competitive NMDA receptor antagonist

Selective mineralcorticoid receptor antagonist

D₂ receptor antagonist

Selective, non-competitive AMPA receptor antagonist

Non-competitive AMPA receptor antagonist. Also blocks kainate GluK3 homomeric receptors.

Dopamine receptor antagonist with partial D₂-like selectivity

Endogenous ionotropic glutamate / nicotinic antagonist.

Novel, potent covalent A_2A antagonist. Binds irreversibly.

Novel, potent, selective A₃AR covalent antagonist