Cannabinoid

Potent, selective μ-opioid receptor agonist

Potent muscarinic acetylcholine receptor superagonist. Also binds the hM3R-miniG_q DREADD receptor.

The first covalent hA₁AR partial agonist. Binds Irreversibly.

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Potent, selective group II receptor agonist

Myelin oligodendrocyte glycoprotein fragment. Induces experimental multiple sclerosis-like disease.

Newly identified, highly selective FFA2-DREADD agonist

Potent GABA_B receptor agonist