Actin

Potent, selective CXCR4 antagonist. Mobilizes hematopoietic stem cells.

Selective PAR₂ peptide antagonist

Dopamine receptor antagonist with partial D₂-like selectivity

Selective, non-peptide AT₁ antagonist

Potent glucocorticoid and progesterone receptor antagonist. Also used for gene editing as a mifepristone inducible Cas9 and Cpf1 CRISPR effector.

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

AT₁ antagonist and PPARγ partial agonist