Receptors & Transporters

Potent, selective µ-opioid receptor agonist

Selective I₂-imidazoline receptor ligand

The first covalent hA₁AR partial agonist. Binds Irreversibly.

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Novel, clickable Adenosine hA₃AR Affinity-Based Probe (AfBP).

Potent, selective group II receptor agonist

Selective H₁ receptor inverse agonist

5-HT₁/5-HT₂ antagonist. Shows affinity for 5-HT₆ and 5-HT₇.

Newly identified, highly selective FFA2-DREADD agonist

5-HT₆ antagonist