CP 465022 hydrochloride product vial image | Hello Bio
CP 465022 hydrochloride product vial image | Hello Bio
Biological Data
Biological description
Potent and non-competitive AMPA receptor antagonist (IC50 = 25 nM). Weakly inhibits NMDA, GABA and kainate receptors. Displays anticonvulsant actions.
This product is a mixture of the active isomer CP 465022 and the inactive isomer CP 465021. The mixture itself is also known as CP 392110.
Please note that there is confusion in the life science marketplace and scientific literature regarding the correct naming of this product and typically, where the product is cited as CP465022, it is generally the mixture of both isomers that is being referred to. If you need any further clarification, please contact customercare@hellobio.com
Solubility & Handling
Solubility overview
Soluble in water (10mM) and in DMSO (100mM)
Storage instructions
Room temperature (desiccate)
Storage of solutions
Prepare and use solutions on the same day if possible. Store solutions at -20°C for up to one month if storage is required. Equilibrate to RT and ensure the solution is precipitate free before use.
Shipping Conditions
Stable for ambient temperature shipping. Follow storage instructions on receipt.
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.
Characterization of the binding site for a novel class of noncompetitive alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor antagonists.
Menniti FS et al (2000) Mol Pharmacol 58(6) : 1310-7.
![CP 465022 hydrochloride [199655-36-2] Chemical Structure](https://cdn.hellobio.com/media/catalog/product//h/b/hb0214.png "CP 465022 hydrochloride [199655-36-2]")
Understanding purity and quality - a guide for life scientists
