Target

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Potent, selective group II receptor agonist

Newly identified, highly selective FFA2-DREADD agonist

TLR1/TLR2 agonist and potent NF-κB activator. Induces cytokine production.

Selective ERα estrogen receptor agonist

Potent GABA_B receptor agonist

Abundant free amino acid found in the brain.

K_ir2.3 channel agonist

Ultrapotent PSEM agonist for PSAM⁴-GlyR and PSAM⁴-5HT3. Brain penetrant.