Target

The first covalent hA₁AR partial agonist. Binds Irreversibly.

Novel, clickable Adenosine hA₁AR Affinity-Based Probe (AfBP).

Novel, clickable Adenosine hA₃AR Affinity-Based Probe (AfBP).

Potent, selective group II receptor agonist

Free fatty acid 1 (FFA₁) receptor agonist

Selective H₁ receptor inverse agonist

5-HT₁/5-HT₂ antagonist. Shows affinity for 5-HT₆ and 5-HT₇.

Newly identified, highly selective FFA2-DREADD agonist

5-HT₆ antagonist

Potent, selective, competitive GABA_A receptor agonist