My Cart
My account
Menu
Main Menu

Arcaine sulfate

(HB0118)
Be the first to add a publication
Technical documents: SDS CoA Datasheet
Be the first to review this product
Add to Wish List

Product overview

Name Arcaine sulfate
Purity >99%
Description Competitive NMDA receptor antagonist / NOS inhibitor
Biological Data Solubility & Handling Chemical Data Related Areas Calculators Technical guides (4) Reviews References (4)
Write Your Own Review
You're reviewing:Arcaine sulfate
Rate this item:

Biological Data

Biological description Competitive NMDA receptor antagonist. Binds at the polyamine site. Also a NOS (Nitric oxide synthase) inhibitor. Reduces NMDA single-channel currents in a voltage-dependent manner.

Solubility & Handling

Solubility overview Soluble in water (25mM)
Storage instructions Room temperature
Storage of solutions Prepare and use solutions on the same day if possible. Store solutions at -20°C for up to one month if storage is required. Equilibrate to RT and ensure the solution is precipitate free before use.
Shipping Conditions Stable for ambient temperature shipping. Follow storage instructions on receipt.
Important This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

Calculators

Molarity

=
x
x
More Info

Dilution

x
=
x
More Info

Chemical Data

Purity >99%
Chemical name N,N'-1,4-Butanediylbisguanidine sulfate
Molecular Weight 270.31
Chemical structure Arcaine sulfate [14923-17-2] Chemical Structure
Molecular Formula C6H16N6.H2SO4
CAS Number 14923-17-2
PubChem identifier 119020
SMILES C(CCN=C(N)N)CN=C(N)N.OS(=O)(=O)O
InChiKey RWTGFMPOODRXIM-UHFFFAOYSA-N

References for Arcaine sulfate

References are publications that support the biological activity of the product

  • Spermine and arcaine block and permeate N-methyl-D-aspartate receptor channels.

    Araneda RC et al (1999) Biophys J 76(6) : 2899-911.
    Read more (PubMedID: 10354418)

  • Investigation of the actions and antagonist activity of some polyamine analogues in vivo.

    Doyle KM et al (1998) Br J Pharmacol 124(2) : 386-90.
    Read more (PubMedID: 9641557)

  • Structure-activity relationships of arginine analogues on nitric oxide synthase activity in the rat brain.

    Yokoi I et al (1994) Neuropharmacology 33(11) : 1261-5.
    Read more (PubMedID: 7532812)

  • Arcaine is a competitive antagonist of the polyamine site on the NMDA receptor.

    Reynolds IJ (1990) Eur J Pharmacol 177(3) : 215-6.
    Read more (PubMedID: 2155812)

4 Item(s)

Related Products
Grouped product items
Order: HB0118
Pack PriceQty
50mg
$88
Competitive NMDA receptor antagonist / NOS inhibitor
Shipping Info

Standard: $35

Hazardous: $35

Shipped on ice: $35

Shipping will be calculated at checkout

Contact Us

Call 609-683-7500
Fax 609-228-4994

customercare-usa@hellobio.com

New Products in this Area

CGP 78608 hydrochloride
HB0187

Selective, competitive GluN1 NMDAR receptor antagonist. Enhances GluN1/3 activation.

Related Products

NBQX disodium salt
Code:
HB0443
Pack:
1mg, 10mg, 50mg, 50mM (add 1ml water), 100mM (add 1ml water)
Price:
$93, $193, $816, $460, $801
(Free trial)
Potent, selective, competitive AMPA receptor antagonist. Disodium salt.
Ro 25-6981 maleate
Code:
HB0554
Pack:
1mg, 10mg, 50mg
Price:
$64, $136, $563
Selective negative allosteric modulator of GluN2B (NR2B) containing NMDARs
D-AP5
Code:
HB0225
Pack:
1mg, 10mg, 50mg, 100mg, 50mM (add 1ml water), 100mM (add 1ml water)
Price:
$45, $116, $495, $685, $161, $289
(Free trial)

Selective, competitive NMDA receptor antagonist. Inhibits NMDAR-synaptic plasticity.