AM 281 is a potent, selective CB1 receptor antagonist / inverse agonist which is selective for CB1 over CB2 receptors (Ki values are 12 nM and 4200 nM respectively). AM 281 modulates locomotor activity and shows neuroprotective actions in septic shock.
Solubility & Handling
Soluble in DMSO (50 mM with heating)
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.