Potent, highly selective α2 adrenoceptor agonist (Ki values are 1.08 and 1750 nM at α2 and α1 receptors, respectively). Active isomer of medetomidine. Shows greater selectivity for α1-adrenoceptors than clonidine and UK14304. Shows various actions such as hypotensive, bradycardic, anxiolytic, hypothermic, sedative and analgesic properties.
Solubility & Handling
Storage instructions
-20°C
Solubility overview
Soluble in water (100 mM), and in DMSO (100 mM)
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use