Potent, selective and competitive P2X receptor antagonist. Selective for P2X1 receptors (IC50 values are 0.3 and 0.7 nM, 0.3, 1.8, 47 and >300 µM for P2X1, P2X1 + 5, P2X2 + 3, P2X3, P2X2 and P2X4 receptors respectively). Also inhibits FGFR3. Shows potential anti-cancer and anti-thrombotic actions.
Solubility & Handling
Solubility overview
Soluble in water
Storage instructions
Room temperature
Storage of solutions
Prepare and use solutions on the same day if possible. Store solutions at -20°C for up to one month if storage is required. Equilibrate to RT and ensure the solution is precipitate free before use.
Shipping Conditions
Stable for ambient temperature shipping. Follow storage instructions on receipt.
Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.