Product overview

Name I-CBP 112
Purity >98%
Description CBP/p300 Bromodomain inhibitor
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Biological Data

Biological description CBP/p300 Bromodomain inhibitor (IC50 values are 170 and 625 nM). Selective over ATAD2, BAZ2B, BRD2, BRD4, PB1, PCAF, PHIP and TRIM24/TIF-1a. Shows accelerated FRAP recovery at 1 µM.

Solubility & Handling

Storage instructions +4°C
Solubility overview Soluble in DMSO (100mM)
Important This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

Calculators

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Chemical Data

Purity >98%
Chemical name 1-[7-(3,4-Dimethoxyphenyl)-9-[[(3S)-1-methylpiperidin-3-yl]methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
Molecular Weight 468.59
Chemical structure I-CBP 112 Chemical Structure
Molecular Formula C27H36N2O5
CAS Number 1640282-31-0
PubChem identifier 90488984
SMILES COC(C(OC)=C1)=CC=C1C2=CC(OC[C@H]3CCCN(C)C3)=C(OCCN(C(CC)=O)C4)C4=C2
InChiKey YKNAKDFZAWQEEO-IBGZPJMESA-N

References for I-CBP 112

References are publications that support the biological activity of the product

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