Product overview

Name Bisindolylmaleimide X
Description Potent, selective PKC inhibitor
Biological description Potent and selective protein kinase C (PKC) inhibitor (IC = 15 nM). Displays selectivity for PKC-α and PKC-β1 over PKC-βII, PKC-γ and PKC-ε (IC50 values are 8, 8, 14, 13, and 39 nM respectively). Also potent CDK2 antagonist (IC50 = 200 nM).
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Solubility & Handling

Important This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

Calculators

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Dilution

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Chemical Data

Chemical name 3-[8-(aminomethyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione, monohydrochloride
Molecular Weight 461
Molecular Formula C26H24N4O2.HCl
CAS Number 145317-11-9