Potent, selective and competitive TRPV1 channel antagonist (IC50 values are 24.5 and 85.6 nM for human and rat TRPV1 respectively). Competitively inhibits capsaicin binding to rat TRPV1. Displays antihyperalgesic effects.
Solubility & Handling
Soluble in DMSO (50mM) or ethanol (100mM)
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.