Mineralocorticoid

Selective mineralcorticoid receptor antagonist

Estrogen receptor (ER) antagonist and high affinity GPER agonist

Potent glucocorticoid and progesterone receptor antagonist. Also used for gene editing as a mifepristone inducible Cas9 and Cpf1 CRISPR effector.

Selective ERα estrogen receptor antagonist

Selective ERβ estrogen receptor antagonist

Mineralocorticoid and androgen receptor antagonist

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9).

Estrogen receptor antagonist/ partial agonist. May be used in genome engineering (e.g. CreER/ CRISPR-Cas9). Citrate salt.

AT₁ antagonist and PPARγ partial agonist