G protein coupled receptors

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G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

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Items 1-10 of 17

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  1. Description:

    Non-selective β-adrenoceptor antagonist. Also a 5-HT1A receptor antagonist.

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $103
    Qty:
  2. Description:

    5-HT1A partial agonist

    Pack:
    10mg
    Price:
    $83
    Qty:
    Pack:
    50mg
    Price:
    $299
    Qty:
  3. Description:

    Selective h5-HT1D antagonist

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $160
    Qty:
    Pack:
    50mg
    Price:
    $598
    Qty:
  4. BRL 54443 (HB1664)

    Description:

    Potent 5-ht1E/1F receptor agonist

    Pack:
    10mg
    Price:
    $146
    Qty:
    Pack:
    50mg
    Price:
    $501
    Qty:
  5. Description:

    Classic 5-HT1A partial agonist

    Purity:

    >99%

    Pack:
    100mg
    Price:
    $77
    Qty:
  6. Pack:
    10mg
    Price:
    $136
    Qty:
    Pack:
    50mg
    Price:
    $557
    Qty:
  7. Description:

    Selective 5-HT1B/1D receptor agonist.

    Purity:

    >99%

    Pack:
    50mg
    Price:
    $832
    Qty:
  8. Ipsapirone (HB1699)

    Description:

    Selective 5-HT1A agonist

    Purity:

    >99%

    Pack:
    10mg
    Price:
    $119
    Qty:
    Pack:
    50mg
    Price:
    $451
    Qty:
  9. Description:

    5-HT1D-preferring receptor antagonist

    Purity:

    >98%

    Pack:
    10mg
    Price:
    $208
    Qty:
    Pack:
    50mg
    Price:
    $681
    Qty:
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