DNA methyltransferase (DNMT)

Shows no COX-2 inhibitory function. Analog of celecoxib.

Reversibly stimulates SERCA Ca²⁺-ATPase. V-ATPase inhibitor.

Potent AChE inhibitor

Potent, selective AMPK inhibitor. Promotes neural hPSCs differentiation and promotes cardiomyocyte differentiation in mESCs.

Cell-permeable, non-competitive dynamin inhibitor

Broad enzyme inhibitor. Inhibits Gq protein signaling.

Ion chelator

Potent adenosine deaminase and PDE2 inhibitor. Supresses spontaneous hESC differentiation. Also maintains pluripotency of hESCs in the absence of exogenous cytokines.

Macrolide antibiotic

Leukocyte elastase inhibitor